cycLex EphA2 Kinase Assay/Inhibitor Screening Kit-Discontinued



This product has been discontinued.

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  1. Holder N., Klein R. Eph receptors and ephrins: effectors of morphogenesis. Development (Camb.), 126: 2033-2044, 1999.
  2. Dodelet V. C., Pasquale E. B. Eph receptors and ephrin ligands: embryogenesis to tumorigenesis. Oncogene, 19: 5614-5619, 2000
  3. Easty D. J., Herlyn M., Bennett D. C. Abnormal protein tyrosine kinase gene expression during melanoma progression and metastasis. Int. J. Cancer, 60: 129-136, 1995.
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  6. Zelinski D., Zantek N., Stewart J., Irizarry A., Kinch M. EphA2 overexpression causes tumorigenesis of mammary epithelial cells. Cancer Res., 61: 2301-2306, 2001.
  7. Walker-Daniels J., Coffman K., Azimi M., Rhim J. S., Bostwick D. G., Snyder P., Kerns B. J., Waters
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  9. Kinch M. S., Moore M. B., Harpole D. H., Jr. Predictive value of the EphA2 receptor tyrosine kinase in lung cancer recurrence and survival. Clin. Cancer Res., 9: 613-618, 2003.
  10. Miyazaki T., Kato H., Fukuchi M., Nakajima M., Kuwano H. EphA2 overexpression correlates with poor prognosis in esophageal squamous cell carcinoma. Int. J. Cancer, 103: 657-663, 2003.
  11. Miao H., Burnett E., Kinch M., Simon E., Wang B. Activation of EphA2 kinase suppresses integrin function and causes focal-adhesion-kinase dephosphorylation. Nat. Cell Biol., 2: 62-69, 2000.
  12. Dohn M., Jiang J., Chen X. Receptor tyrosine kinase EphA2 is regulated by p53-family proteins and induces apoptosis. Oncogene, 20: 6503-6515, 2001.
  13. Ogawa K., Pasqualini R., Lindberg R., Kain R., Freeman A., Pasquale E. The ephrin-A1 ligand and its receptor, EphA2 are expressed during tumor neovascularization. Oncogene, 19: 6043-6052, 2000.
  14. Hess A. R., Seftor E. A., Gardner L. M., Carles-Kinch K., Schneider G. B., Seftor R. E., Kinch M. S., Hendrix M. J. Molecular regulation of tumor cell vasculogenic mimicry by tyrosine phosphorylation: role of epithelial cell kinase (Eck/EphA2). Cancer Res., 61: 3250-3255, 2001.
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